Assay Detail
Binding
CHEMBL3269020
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Inhibition of Mycobacterium smegmatis MenA
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mycolicibacterium smegmatis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Multitarget drug discovery for tuberculosis and other infectious diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 12 | 5.27 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3261880 | — | — | 1 | 5.40 |
| CHEMBL561057 | SQ109 | 2.0 | 1 | 5.32 |
| CHEMBL3261890 | — | — | 1 | 5.10 |
| CHEMBL3261881 | — | — | 1 | - |
| CHEMBL3261882 | — | — | 1 | - |
| CHEMBL3261883 | — | — | 1 | - |
| CHEMBL3261884 | — | — | 1 | - |
| CHEMBL3261885 | — | — | 1 | - |
| CHEMBL3261886 | — | — | 1 | - |
| CHEMBL3261887 | — | — | 1 | - |
| CHEMBL3261888 | — | — | 1 | - |
| CHEMBL3261889 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3261880 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL561057 | SQ109 | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL3261890 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL3261881 | — | IC50 | - | — | - | |
| CHEMBL3261882 | — | IC50 | - | — | - | |
| CHEMBL3261883 | — | IC50 | - | — | - | |
| CHEMBL3261884 | — | IC50 | - | — | - | |
| CHEMBL3261885 | — | IC50 | - | — | - | |
| CHEMBL3261886 | — | IC50 | - | — | - | |
| CHEMBL3261887 | — | IC50 | - | — | - | |
| CHEMBL3261888 | — | IC50 | - | — | - | |
| CHEMBL3261889 | — | IC50 | - | — | - |