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Assay Detail

CHEMBL3270671

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anticancer activity against human SH-SY5Y cells assessed as reduction in cell viability
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SH-SY5Y
Confidence 1 — Organism
Curated By Autocuration

Target

SH-SY5Y (CHEMBL614910)
Type CELL-LINE
Organism Homo sapiens

Publication

Indirubin core structure of glycogen synthase kinase-3 inhibitors as novel chemotype for intervention with 5-lipoxygenase.
Pergola C, Gaboriaud-Kolar N, Jestädt N, König S, Kritsanida M, Schaible AM, Li H, Garscha U, Weinigel C, Barz D, Albring KF, Huber O, Skaltsounis AL, Werz O.
J Med Chem (2014) 57 : 3715 -3723
PubMed 24697244 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.10 5.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1092509 1 5.10
CHEMBL409450 6BIO 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1092509 EC50 = 8000.0 nM 5.10
CHEMBL409450 6BIO EC50 > 30000.0 nM -