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Assay Detail

CHEMBL3362076

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of his-tagged active RSK2 (unknown origin) expressed in Sf9 cells after 10 to 45 mins by ELISA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type Sf9
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Ribosomal protein S6 kinase alpha-3 (CHEMBL2345)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Kaempferol, a potential cytostatic and cure for inflammatory disorders.
Rajendran P, Rengarajan T, Nandakumar N, Palaniswami R, Nishigaki Y, Nishigaki I.
Eur J Med Chem (2014) 86 : 103 -112
PubMed 25147152 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.05 7.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL240954 1 7.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL240954 IC50 = 89.0 nM 7.05