Assay Detail
Binding
CHEMBL3367178
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Inhibition of AP-1 bZIP domain DNA binding activity (unknown origin) by ELISA
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Small molecule inhibitors targeting activator protein 1 (AP-1).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.60 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3222137 | — | — | 1 | 5.00 |
| CHEMBL3222140 | — | — | 1 | 4.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3222137 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL3222140 | — | IC50 | = | 64000.0 | nM | 4.19 |