Assay Detail
Binding
CHEMBL3367259
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to benzodiazepine receptor (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Target
Benzodiazepine receptors; peripheral & central (CHEMBL2096683) ↗| Type | SELECTIVITY GROUP |
| Organism | Rattus norvegicus |
Publication
Flavones: an important scaffold for medicinal chemistry.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.90 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL335086 | — | — | 1 | 9.05 |
| CHEMBL54341 | — | — | 1 | 8.82 |
| CHEMBL292868 | — | — | 1 | 8.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL335086 | — | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL54341 | — | Ki | = | 1.5 | nM | 8.82 |
| CHEMBL292868 | — | Ki | = | 1.5 | nM | 8.82 |