Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3372608

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of IFN-gamma/LPS-induced PGE2 production in mouse RAW264.7 cells after 17 to 20 hrs by EIA method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Inhibition of prostaglandin E(2) production by synthetic minor prenylated chalcones and flavonoids: synthesis, biological activity, crystal structure, and in silico evaluation.
Rullah K, Mohd Aluwi MF, Yamin BM, Abdul Bahari MN, Wei LS, Ahmad S, Abas F, Ismail NH, Jantan I, Wai LK.
Bioorg Med Chem Lett (2014) 24 : 3826 -3834
PubMed 25027933 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.34 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7162 NS-398 1 7.00
CHEMBL3318159 1 5.68

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7162 NS-398 IC50 = 100.0 nM 7.00
CHEMBL3318159 IC50 = 2100.0 nM 5.68