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Assay Detail

CHEMBL3373164

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Escherichia coli GyrB A2B2 subunits assessed reduction in DNA supercoiling activity by malachite green dye based by spectrophotometry
50
Total Activities
50
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Escherichia coli
Confidence 7 — Homologous single protein target
Curated By Autocuration

Target

DNA gyrase (CHEMBL2094139)
Type PROTEIN COMPLEX
Organism Escherichia coli

Publication

Pyridine-3-carboxamide-6-yl-ureas as novel inhibitors of bacterial DNA gyrase: structure based design, synthesis, SAR and antimicrobial activity.
Yule IA, Czaplewski LG, Pommier S, Davies DT, Narramore SK, Fishwick CW.
Eur J Med Chem (2014) 86 : 31 -38
PubMed 25137573 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 50 5.88 7.55

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3329317 1 7.55
CHEMBL3329318 1 7.44
CHEMBL3329312 1 7.41
CHEMBL3329307 1 7.40
CHEMBL3329319 1 7.34
CHEMBL3329316 1 7.03
CHEMBL3329292 1 7.01
CHEMBL3329291 1 7.00
CHEMBL3329311 1 6.96
CHEMBL3329308 1 6.85
CHEMBL3329313 1 6.82
CHEMBL3329309 1 6.82
CHEMBL3329310 1 6.77
CHEMBL3329287 1 6.38
CHEMBL3329221 1 6.37
CHEMBL3329297 1 6.26
CHEMBL3329298 1 6.25
CHEMBL3329305 1 6.18
CHEMBL3329302 1 6.09
CHEMBL3329288 1 6.02
CHEMBL3329299 1 5.95
CHEMBL3329274 1 5.80
CHEMBL3329314 1 5.70
CHEMBL3329275 1 5.68
CHEMBL3329304 1 5.67
CHEMBL3329303 1 5.53
CHEMBL3329277 1 5.52
CHEMBL3329300 1 5.52
CHEMBL3329276 1 5.48
CHEMBL3329278 1 5.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3329317 IC50 = 28.0 nM 7.55
CHEMBL3329318 IC50 = 36.0 nM 7.44
CHEMBL3329312 IC50 = 39.0 nM 7.41
CHEMBL3329307 IC50 = 40.0 nM 7.40
CHEMBL3329319 IC50 = 46.0 nM 7.34
CHEMBL3329316 IC50 = 93.0 nM 7.03
CHEMBL3329292 IC50 = 98.0 nM 7.01
CHEMBL3329291 IC50 = 99.0 nM 7.00
CHEMBL3329311 IC50 = 110.0 nM 6.96
CHEMBL3329308 IC50 = 140.0 nM 6.85
CHEMBL3329313 IC50 = 150.0 nM 6.82
CHEMBL3329309 IC50 = 150.0 nM 6.82
CHEMBL3329310 IC50 = 170.0 nM 6.77
CHEMBL3329287 IC50 = 420.0 nM 6.38
CHEMBL3329221 IC50 = 430.0 nM 6.37
CHEMBL3329297 IC50 = 550.0 nM 6.26
CHEMBL3329298 IC50 = 560.0 nM 6.25
CHEMBL3329305 IC50 = 660.0 nM 6.18
CHEMBL3329302 IC50 = 810.0 nM 6.09
CHEMBL3329288 IC50 = 960.0 nM 6.02
CHEMBL3329299 IC50 = 1130.0 nM 5.95
CHEMBL3329274 IC50 = 1600.0 nM 5.80
CHEMBL3329314 IC50 = 2000.0 nM 5.70
CHEMBL3329275 IC50 = 2100.0 nM 5.68
CHEMBL3329304 IC50 = 2120.0 nM 5.67
CHEMBL3329303 IC50 = 2960.0 nM 5.53
CHEMBL3329300 IC50 = 3020.0 nM 5.52
CHEMBL3329277 IC50 = 3000.0 nM 5.52
CHEMBL3329276 IC50 = 3300.0 nM 5.48
CHEMBL3329278 IC50 = 3400.0 nM 5.47
CHEMBL3329284 IC50 = 3500.0 nM 5.46
CHEMBL3329279 IC50 = 3800.0 nM 5.42
CHEMBL3329306 IC50 = 4810.0 nM 5.32
CHEMBL3329315 IC50 = 4900.0 nM 5.31
CHEMBL3329293 IC50 = 5140.0 nM 5.29
CHEMBL3329285 IC50 = 5300.0 nM 5.28
CHEMBL3329294 IC50 = 5660.0 nM 5.25
CHEMBL3329272 IC50 = 6000.0 nM 5.22
CHEMBL3329282 IC50 = 6200.0 nM 5.21
CHEMBL3329301 IC50 = 7270.0 nM 5.14
CHEMBL3329283 IC50 = 7500.0 nM 5.12
CHEMBL3329273 IC50 = 7700.0 nM 5.11
CHEMBL3706672 IC50 = 8400.0 nM 5.08
CHEMBL3329286 IC50 = 14000.0 nM 4.85
CHEMBL3329295 IC50 = 18000.0 nM 4.75
CHEMBL3329289 IC50 = 23100.0 nM 4.64
CHEMBL3329280 IC50 = 24500.0 nM 4.61
CHEMBL3329296 IC50 = 33200.0 nM 4.48
CHEMBL3329281 IC50 = 40400.0 nM 4.39
CHEMBL3094347 IC50 < 750.0 nM -