Assay Detail
Functional
CHEMBL3374386
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human OVCAR5 cells after 48 hrs by MTT assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OVCAR-5 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
An investigation of in vitro cytotoxicity and apoptotic potential of aromatic diselenides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 4.57 | 4.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3314697 | — | — | 1 | 4.80 |
| CHEMBL3314693 | — | — | 1 | 4.70 |
| CHEMBL3314696 | — | — | 1 | 4.68 |
| CHEMBL3314695 | — | — | 1 | 4.62 |
| CHEMBL3314698 | — | — | 1 | 4.60 |
| CHEMBL2409555 | — | — | 1 | 4.58 |
| CHEMBL3314689 | — | — | 1 | 4.57 |
| CHEMBL3314694 | — | — | 1 | 4.57 |
| CHEMBL2002452 | — | — | 1 | 4.51 |
| CHEMBL3314692 | — | — | 1 | 4.47 |
| CHEMBL3122204 | — | — | 1 | 4.42 |
| CHEMBL3314690 | — | — | 1 | 4.42 |
| CHEMBL3314691 | — | — | 1 | 4.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3314697 | — | IC50 | = | 16000.0 | nM | 4.80 |
| CHEMBL3314693 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL3314696 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL3314695 | — | IC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL3314698 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL2409555 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL3314689 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL3314694 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL2002452 | — | IC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL3314692 | — | IC50 | = | 34000.0 | nM | 4.47 |
| CHEMBL3122204 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL3314690 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL3314691 | — | IC50 | = | 39000.0 | nM | 4.41 |