Assay Detail
Functional
CHEMBL3374387
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Cytotoxicity against human 786-O cells after 48 hrs by MTT assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | 786-0 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
An investigation of in vitro cytotoxicity and apoptotic potential of aromatic diselenides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 4.51 | 4.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3314693 | — | — | 1 | 4.62 |
| CHEMBL3314696 | — | — | 1 | 4.57 |
| CHEMBL3314697 | — | — | 1 | 4.57 |
| CHEMBL2409555 | — | — | 1 | 4.55 |
| CHEMBL3314689 | — | — | 1 | 4.54 |
| CHEMBL2002452 | — | — | 1 | 4.54 |
| CHEMBL3314695 | — | — | 1 | 4.52 |
| CHEMBL3314698 | — | — | 1 | 4.50 |
| CHEMBL3314692 | — | — | 1 | 4.48 |
| CHEMBL3314694 | — | — | 1 | 4.48 |
| CHEMBL3122204 | — | — | 1 | 4.42 |
| CHEMBL3314691 | — | — | 1 | 4.40 |
| CHEMBL3314690 | — | — | 1 | 4.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3314693 | — | IC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL3314696 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL3314697 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL2409555 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL3314689 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL2002452 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL3314695 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL3314698 | — | IC50 | = | 32000.0 | nM | 4.50 |
| CHEMBL3314692 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL3314694 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL3122204 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL3314691 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL3314690 | — | IC50 | = | 42000.0 | nM | 4.38 |