Assay Detail
Binding
CHEMBL3375012
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]GR100679 from NK2 receptor (unknown origin) expressed in CHO/T cells
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO/T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Toward fluorescent probes for G-protein-coupled receptors (GPCRs).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 9 | 8.45 | 9.81 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2370064 | — | — | 1 | 9.81 |
| CHEMBL217406 | NEUROKININ A | — | 1 | 8.92 |
| CHEMBL3360196 | — | — | 1 | 8.87 |
| CHEMBL3360197 | — | — | 1 | 8.84 |
| CHEMBL3360198 | — | — | 1 | 8.83 |
| CHEMBL3360199 | — | — | 1 | 8.80 |
| CHEMBL3360201 | — | — | 1 | 8.23 |
| CHEMBL3360200 | — | — | 1 | 8.08 |
| CHEMBL3360202 | — | — | 1 | 5.71 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2370064 | — | Ki | = | 0.1549 | nM | 9.81 |
| CHEMBL217406 | NEUROKININ A | Ki | = | 1.202 | nM | 8.92 |
| CHEMBL3360196 | — | Ki | = | 1.349 | nM | 8.87 |
| CHEMBL3360197 | — | Ki | = | 1.445 | nM | 8.84 |
| CHEMBL3360198 | — | Ki | = | 1.479 | nM | 8.83 |
| CHEMBL3360199 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL3360201 | — | Ki | = | 5.888 | nM | 8.23 |
| CHEMBL3360200 | — | Ki | = | 8.318 | nM | 8.08 |
| CHEMBL3360202 | — | Ki | = | 1949.84 | nM | 5.71 |