Assay Detail
Binding
CHEMBL3378403
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Inhibition of FAAH, TRPV1, and COX2 by NSAID-serotonin conjugates.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.97 | 5.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3359452 | — | — | 1 | 5.30 |
| CHEMBL3359453 | — | — | 1 | 4.82 |
| CHEMBL191534 | — | — | 1 | 4.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3359452 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL3359453 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL191534 | — | IC50 | = | 16000.0 | nM | 4.80 |