Assay Detail
Binding
CHEMBL3378639
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]SS-14 from human SSTR3 expressed in CHO cells by TopCount analyzer
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 8.28 | 9.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3323074 | — | — | 1 | 9.19 |
| CHEMBL3323076 | — | — | 1 | 9.11 |
| CHEMBL3323072 | — | — | 1 | 9.08 |
| CHEMBL3323084 | — | — | 1 | 8.91 |
| CHEMBL3323073 | — | — | 1 | 8.82 |
| CHEMBL3323078 | — | — | 1 | 8.76 |
| CHEMBL3323082 | — | — | 1 | 8.67 |
| CHEMBL3323079 | — | — | 1 | 8.54 |
| CHEMBL3323077 | — | — | 1 | 8.47 |
| CHEMBL3323080 | — | — | 1 | 8.36 |
| CHEMBL3323075 | — | — | 1 | 8.31 |
| CHEMBL3323085 | — | — | 1 | 7.97 |
| CHEMBL3323086 | — | — | 1 | 7.62 |
| CHEMBL3323083 | — | — | 1 | 7.14 |
| CHEMBL3323081 | — | — | 1 | 7.13 |
| CHEMBL3323087 | — | — | 1 | 6.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3323074 | — | IC50 | = | 0.64 | nM | 9.19 |
| CHEMBL3323076 | — | IC50 | = | 0.78 | nM | 9.11 |
| CHEMBL3323072 | — | IC50 | = | 0.83 | nM | 9.08 |
| CHEMBL3323084 | — | IC50 | = | 1.22 | nM | 8.91 |
| CHEMBL3323073 | — | IC50 | = | 1.52 | nM | 8.82 |
| CHEMBL3323078 | — | IC50 | = | 1.72 | nM | 8.76 |
| CHEMBL3323082 | — | IC50 | = | 2.13 | nM | 8.67 |
| CHEMBL3323079 | — | IC50 | = | 2.91 | nM | 8.54 |
| CHEMBL3323077 | — | IC50 | = | 3.36 | nM | 8.47 |
| CHEMBL3323080 | — | IC50 | = | 4.41 | nM | 8.36 |
| CHEMBL3323075 | — | IC50 | = | 4.87 | nM | 8.31 |
| CHEMBL3323085 | — | IC50 | = | 10.8 | nM | 7.97 |
| CHEMBL3323086 | — | IC50 | = | 23.7 | nM | 7.62 |
| CHEMBL3323083 | — | IC50 | = | 72.7 | nM | 7.14 |
| CHEMBL3323081 | — | IC50 | = | 74.7 | nM | 7.13 |
| CHEMBL3323087 | — | IC50 | = | 409.0 | nM | 6.39 |