Assay Detail
Binding
CHEMBL3387052
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Inhibition of human recombinant COX2 pre-incubated for 15 mins before arachidonic acid addition by fluorescence micro plate reader method
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Bioactive compounds from the insect Aspongopus chinensis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 4.85 | 5.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3338322 | — | — | 1 | 5.19 |
| CHEMBL137743 | — | — | 1 | 4.72 |
| CHEMBL75390 | — | — | 1 | 4.65 |
| CHEMBL3338324 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3338322 | — | IC50 | = | 6500.0 | nM | 5.19 |
| CHEMBL137743 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL75390 | — | IC50 | = | 22200.0 | nM | 4.65 |
| CHEMBL3338324 | — | IC50 | = | 117000.0 | nM | - |