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Assay Detail

CHEMBL3390168

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of LPS and IFNgamma-induced nitric oxide production in mouse RAW264.7 cells incubated for 16 hrs by Griess assay
11
Total Activities
11
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Polyyne hybrid compounds from Notopterygium incisum with peroxisome proliferator-activated receptor gamma agonistic effects.
Liu X, Kunert O, Blunder M, Fakhrudin N, Noha SM, Malainer C, Schinkovitz A, Heiss EH, Atanasov AG, Kollroser M, Schuster D, Dirsch VM, Bauer R.
J Nat Prod (2014) 77 : 2513 -2521
PubMed 25333853 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Inhibition 10 - -
IC50 1 4.84 4.84

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3358036 1 4.84
CHEMBL3358033 1 -
CHEMBL3358034 1 -
CHEMBL3358035 1 -
CHEMBL3358037 1 -
CHEMBL3358038 1 -
CHEMBL3358039 1 -
CHEMBL3358040 1 -
CHEMBL3358041 1 -
CHEMBL3358042 1 -
CHEMBL3358043 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3358036 IC50 = 14600.0 nM 4.84
CHEMBL3358033 Inhibition - % -
CHEMBL3358034 Inhibition - % -
CHEMBL3358035 Inhibition - % -
CHEMBL3358037 Inhibition - % -
CHEMBL3358038 Inhibition - % -
CHEMBL3358039 Inhibition - % -
CHEMBL3358040 Inhibition - % -
CHEMBL3358041 Inhibition - % -
CHEMBL3358042 Inhibition - % -
CHEMBL3358043 Inhibition - % -