Assay Detail
Binding
CHEMBL3391163
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Inhibition of AmpC beta-lactamase (unknown origin)
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Not specified |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Boronic acids in medicinal chemistry: anticancer, antibacterial and antiviral applications
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 7.69 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL429972 | — | — | 1 | 9.00 |
| CHEMBL257468 | — | — | 1 | 9.00 |
| CHEMBL404155 | — | — | 1 | 7.46 |
| CHEMBL617 | CEPHALOTHIN | 4.0 | 1 | 6.50 |
| CHEMBL3347545 | — | — | 1 | 6.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL429972 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL257468 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL404155 | — | Ki | = | 35.0 | nM | 7.46 |
| CHEMBL617 | CEPHALOTHIN | Ki | = | 320.0 | nM | 6.50 |
| CHEMBL3347545 | — | Ki | = | 320.0 | nM | 6.50 |