Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3396046

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against rat C6 cells assessed as reduction in cell viability at 0.1 to 5 uM after 24 hrs by MTT assay
4
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Cell Type C6
Confidence 1 — Organism
Curated By Autocuration

Target

C6 (CHEMBL614657)
Type CELL-LINE
Organism Rattus norvegicus

Publication

Haloperidol metabolite II prodrug: asymmetric synthesis and biological evaluation on rat C6 glioma cells.
Sozio P, Fiorito J, Di Giacomo V, Di Stefano A, Marinelli L, Cacciatore I, Cataldi A, Pacella S, Turkez H, Parenti C, Rescifina A, Marrazzo A.
Eur J Med Chem (2015) 90 : 1 -9
PubMed 25461306 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Activity 3 - -
IC50 1 5.30 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1649601 2 5.30
CHEMBL3393790 1 -
CHEMBL3393789 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1649601 IC50 = 5000.0 nM 5.30
CHEMBL3393790 Activity - -
CHEMBL3393789 Activity - -
CHEMBL1649601 Activity - -