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Assay Detail

CHEMBL3406549

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of tyrosinase (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Tyrosinase (CHEMBL1973)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Effect of the tyrosinase inhibitor (S)-N-trans-feruloyloctopamine from garlic skin on tyrosinase gene expression and melanine accumulation in melanoma cells.
Wu Y, Wu ZR, Chen P, Yang-Li, Deng WR, Wang YQ, Li HY.
Bioorg Med Chem Lett (2015) 25 : 1476 -1478
PubMed 25726329 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.38 4.49

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL196 ASCORBIC ACID 4.0 1 4.49
CHEMBL242080 E319 1 4.27

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL196 ASCORBIC ACID IC50 = 32500.0 nM 4.49
CHEMBL242080 E319 IC50 = 54200.0 nM 4.27