Assay Detail
Binding
CHEMBL3411253
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human KLF10 expressed in human HeLa cells assessed as reduction in transcriptional activity after 24 hrs by CACCC-responsive promoter driven TK-luciferase reporter gene assay
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HeLa |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of small molecule inhibitors to Krüppel-like factor 10 (KLF10): implications for modulation of T regulatory cell differentiation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 31 | 4.35 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1333704 | — | — | 1 | 5.00 |
| CHEMBL3410747 | — | — | 1 | 4.40 |
| CHEMBL2179992 | — | — | 1 | 4.37 |
| CHEMBL1324 | TOLCAPONE | 4.0 | 1 | 4.30 |
| CHEMBL641 | ATOMOXETINE | 4.0 | 1 | 4.00 |
| CHEMBL3410732 | — | — | 1 | 4.00 |
| CHEMBL3410741 | — | — | 1 | - |
| CHEMBL3410739 | — | — | 1 | - |
| CHEMBL3410640 | — | — | 1 | - |
| CHEMBL1407890 | — | — | 1 | - |
| CHEMBL3410731 | — | — | 1 | - |
| CHEMBL3410733 | — | — | 1 | - |
| CHEMBL3410734 | — | — | 1 | - |
| CHEMBL3410735 | — | — | 1 | - |
| CHEMBL490514 | — | — | 1 | - |
| CHEMBL3410736 | — | — | 1 | - |
| CHEMBL3410737 | — | — | 1 | - |
| CHEMBL3410738 | — | — | 1 | - |
| CHEMBL1487891 | — | — | 1 | - |
| CHEMBL1350093 | — | — | 1 | - |
| CHEMBL1419342 | — | — | 1 | - |
| CHEMBL592869 | — | — | 1 | - |
| CHEMBL3410749 | — | — | 1 | - |
| CHEMBL3410641 | — | — | 1 | - |
| CHEMBL3410746 | — | — | 1 | - |
| CHEMBL3410745 | — | — | 1 | - |
| CHEMBL3410744 | — | — | 1 | - |
| CHEMBL3410743 | — | — | 1 | - |
| CHEMBL3410742 | — | — | 1 | - |
| CHEMBL3410748 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1333704 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL3410747 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL2179992 | — | IC50 | = | 43000.0 | nM | 4.37 |
| CHEMBL1324 | TOLCAPONE | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL641 | ATOMOXETINE | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL3410732 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL3410640 | — | IC50 | - | — | - | |
| CHEMBL3410740 | — | IC50 | - | — | - | |
| CHEMBL1407890 | — | IC50 | - | — | - | |
| CHEMBL3410731 | — | IC50 | - | — | - | |
| CHEMBL3410733 | — | IC50 | - | — | - | |
| CHEMBL3410734 | — | IC50 | - | — | - | |
| CHEMBL3410735 | — | IC50 | - | — | - | |
| CHEMBL490514 | — | IC50 | = | 200000.0 | nM | - |
| CHEMBL3410736 | — | IC50 | - | — | - | |
| CHEMBL3410737 | — | IC50 | - | — | - | |
| CHEMBL3410738 | — | IC50 | - | — | - | |
| CHEMBL3410739 | — | IC50 | - | — | - | |
| CHEMBL3410741 | — | IC50 | - | — | - | |
| CHEMBL1487891 | — | IC50 | - | — | - | |
| CHEMBL1350093 | — | IC50 | - | — | - | |
| CHEMBL1419342 | — | IC50 | - | — | - | |
| CHEMBL592869 | — | IC50 | - | — | - | |
| CHEMBL3410749 | — | IC50 | - | — | - | |
| CHEMBL3410641 | — | IC50 | = | 112000.0 | nM | - |
| CHEMBL3410746 | — | IC50 | - | — | - | |
| CHEMBL3410745 | — | IC50 | - | — | - | |
| CHEMBL3410744 | — | IC50 | - | — | - | |
| CHEMBL3410743 | — | IC50 | - | — | - | |
| CHEMBL3410742 | — | IC50 | - | — | - | |
| CHEMBL3410748 | — | IC50 | - | — | - |