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Assay Detail

CHEMBL3414018

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human carbonic anhydrase 1
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Carbonic anhydrase 1 (CHEMBL261)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

1,3,4-Thiadiazoles: a potent multi targeted pharmacological scaffold.
Haider S, Alam MS, Hamid H.
Eur J Med Chem (2015) 92 : 156 -177
PubMed 25553540 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.52 8.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3408993 1 8.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3408993 Ki = 3.0 nM 8.52