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Assay Detail

CHEMBL3418917

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HIV-1 3B infected in human HeLa-CD4-LTR-beta-gal cells after 1 day by spectroscopic analysis
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Confidence 1 — Organism
Curated By Autocuration

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domain.
Cuzzucoli Crucitti G, Métifiot M, Pescatori L, Messore A, Madia VN, Pupo G, Saccoliti F, Scipione L, Tortorella S, Esposito F, Corona A, Cadeddu M, Marchand C, Pommier Y, Tramontano E, Costi R, Di Santo R.
J Med Chem (2015) 58 : 1915 -1928
PubMed 25629256 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 26 5.58 7.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL254316 RALTEGRAVIR 4.0 1 7.80
CHEMBL3415832 1 6.25
CHEMBL3415845 1 6.24
CHEMBL3415846 1 6.20
CHEMBL3415843 1 6.18
CHEMBL3415853 1 6.16
CHEMBL3415842 1 6.16
CHEMBL3415833 1 6.05
CHEMBL499273 1 6.00
CHEMBL3415841 1 5.92
CHEMBL3415856 1 5.70
CHEMBL3238122 1 5.44
CHEMBL3415840 1 5.37
CHEMBL3415852 1 4.76
CHEMBL3415835 1 4.72
CHEMBL3415834 1 4.72
CHEMBL3415836 1 4.70
CHEMBL3415854 1 4.69
CHEMBL3415837 1 4.32
CHEMBL3415839 1 4.30
CHEMBL3415847 1 -
CHEMBL3415848 1 -
CHEMBL3415851 1 -
CHEMBL557770 1 -
CHEMBL3415855 1 -
CHEMBL3415844 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL254316 RALTEGRAVIR EC50 = 16.0 nM 7.80
CHEMBL3415832 EC50 = 560.0 nM 6.25
CHEMBL3415845 EC50 = 580.0 nM 6.24
CHEMBL3415846 EC50 = 630.0 nM 6.20
CHEMBL3415843 EC50 = 660.0 nM 6.18
CHEMBL3415853 EC50 = 700.0 nM 6.16
CHEMBL3415842 EC50 = 700.0 nM 6.16
CHEMBL3415833 EC50 = 900.0 nM 6.05
CHEMBL499273 EC50 = 1000.0 nM 6.00
CHEMBL3415841 EC50 = 1200.0 nM 5.92
CHEMBL3415856 EC50 = 2000.0 nM 5.70
CHEMBL3238122 EC50 = 3600.0 nM 5.44
CHEMBL3415840 EC50 = 4300.0 nM 5.37
CHEMBL3415852 EC50 = 17200.0 nM 4.76
CHEMBL3415835 EC50 = 19000.0 nM 4.72
CHEMBL3415834 EC50 = 19000.0 nM 4.72
CHEMBL3415836 EC50 = 20000.0 nM 4.70
CHEMBL3415854 EC50 = 20400.0 nM 4.69
CHEMBL3415837 EC50 = 48000.0 nM 4.32
CHEMBL3415839 EC50 = 50000.0 nM 4.30
CHEMBL3415847 EC50 > 50000.0 nM -
CHEMBL3415848 EC50 > 50000.0 nM -
CHEMBL3415851 EC50 > 50000.0 nM -
CHEMBL557770 EC50 > 50000.0 nM -
CHEMBL3415855 EC50 < 200.0 nM -
CHEMBL3415844 EC50 > 50000.0 nM -