Assay Detail
Binding
CHEMBL3419155
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive binding affinity to human MAP3K2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mitogen-activated protein kinase kinase kinase 2 (CHEMBL5914) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery and profiling of a selective and efficacious Syk inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.85 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3416026 | — | — | 1 | 6.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3416026 | — | Kd | = | 140.0 | nM | 6.85 |