Assay Detail
Binding
CHEMBL3419227
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to BAZ2B (unknown origin) by isothermal titration calorimetric analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Bromodomain adjacent to zinc finger domain protein 2B (CHEMBL1741220) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Structure enabled design of BAZ2-ICR, a chemical probe targeting the bromodomains of BAZ2A and BAZ2B.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.77 | 6.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4296718 | — | — | 1 | 6.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4296718 | — | Kd | = | 170.0 | nM | 6.77 |