Assay Detail
Functional
CHEMBL3429703
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Antiviral activity in HCV 1b infected in HUH 7-lunet cells after 3 days by Dual-Glo luciferase assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Hepacivirus hominis |
| Cell Type | HUH 7-lunet |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 6.26 | 7.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3426601 | — | — | 1 | 7.06 |
| CHEMBL3426603 | — | — | 1 | 6.68 |
| CHEMBL236207 | BETA-2'-C-METHYL-7-DEAZA-ADENOSINE | — | 1 | 6.68 |
| CHEMBL3426599 | — | — | 1 | 6.54 |
| CHEMBL3426602 | — | — | 1 | 6.44 |
| CHEMBL3426598 | — | — | 1 | 6.43 |
| CHEMBL3426596 | — | — | 1 | 6.04 |
| CHEMBL3426597 | — | — | 1 | 6.02 |
| CHEMBL3426594 | — | — | 1 | 5.99 |
| CHEMBL2397317 | — | — | 1 | 5.99 |
| CHEMBL3426595 | — | — | 1 | 5.92 |
| CHEMBL3426600 | — | — | 1 | 5.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3426601 | — | EC50 | = | 87.0 | nM | 7.06 |
| CHEMBL3426603 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL236207 | BETA-2'-C-METHYL-7-DEAZA-ADENOSINE | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL3426599 | — | EC50 | = | 290.0 | nM | 6.54 |
| CHEMBL3426602 | — | EC50 | = | 360.0 | nM | 6.44 |
| CHEMBL3426598 | — | EC50 | = | 370.0 | nM | 6.43 |
| CHEMBL3426596 | — | EC50 | = | 910.0 | nM | 6.04 |
| CHEMBL3426597 | — | EC50 | = | 960.0 | nM | 6.02 |
| CHEMBL3426594 | — | EC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL2397317 | — | EC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL3426595 | — | EC50 | = | 1210.0 | nM | 5.92 |
| CHEMBL3426600 | — | EC50 | = | 5300.0 | nM | 5.28 |