Assay Detail
Functional
CHEMBL3429704
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Antiviral activity in HCV 2a JFH1 infected in HUH 7-lunet cells after 3 days by Dual-Glo luciferase assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Hepacivirus hominis |
| Cell Type | HUH 7-lunet |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 4.91 | 6.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL236207 | BETA-2'-C-METHYL-7-DEAZA-ADENOSINE | — | 1 | 6.68 |
| CHEMBL3426601 | — | — | 1 | 4.97 |
| CHEMBL3426600 | — | — | 1 | 4.87 |
| CHEMBL3426598 | — | — | 1 | 4.75 |
| CHEMBL3426603 | — | — | 1 | 4.58 |
| CHEMBL3426602 | — | — | 1 | 4.55 |
| CHEMBL3426599 | — | — | 1 | 4.50 |
| CHEMBL3426596 | — | — | 1 | 4.37 |
| CHEMBL3426594 | — | — | 1 | - |
| CHEMBL3426595 | — | — | 1 | - |
| CHEMBL3426597 | — | — | 1 | - |
| CHEMBL2397317 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL236207 | BETA-2'-C-METHYL-7-DEAZA-ADENOSINE | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL3426601 | — | EC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL3426600 | — | EC50 | = | 13600.0 | nM | 4.87 |
| CHEMBL3426598 | — | EC50 | = | 17900.0 | nM | 4.75 |
| CHEMBL3426603 | — | EC50 | = | 26500.0 | nM | 4.58 |
| CHEMBL3426602 | — | EC50 | = | 27900.0 | nM | 4.55 |
| CHEMBL3426599 | — | EC50 | = | 31800.0 | nM | 4.50 |
| CHEMBL3426596 | — | EC50 | = | 42500.0 | nM | 4.37 |
| CHEMBL3426594 | — | EC50 | > | 44000.0 | nM | - |
| CHEMBL3426595 | — | EC50 | > | 44000.0 | nM | - |
| CHEMBL3426597 | — | EC50 | > | 44000.0 | nM | - |
| CHEMBL2397317 | — | EC50 | > | 44000.0 | nM | - |