Assay Detail
Functional
CHEMBL3562038
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. SNU-C1 viability from Cell TiterGlo-IC50. (Class of assay: confirmatory)
230
Total Activities
229
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | SNU-C1 |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 230 | 6.13 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 9.00 |
| CHEMBL232201 | BENZIODARONE | 4.0 | 1 | 9.00 |
| CHEMBL24944 | TRIBROMSALAN | 4.0 | 1 | 9.00 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 8.83 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 8.64 |
| CHEMBL3559830 | — | — | 1 | 8.49 |
| CHEMBL1375045 | — | — | 1 | 8.40 |
| CHEMBL5219790 | CETRIMIDE | 2.0 | 1 | 8.29 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 8.06 |
| CHEMBL1981438 | CLOFLUCARBAN | 2.0 | 1 | 8.05 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 7.84 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 7.77 |
| CHEMBL81782 | — | — | 1 | 7.76 |
| CHEMBL2355417 | — | — | 1 | 7.70 |
| CHEMBL2361697 | — | — | 1 | 7.53 |
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 7.50 |
| CHEMBL1545634 | — | — | 1 | 7.45 |
| CHEMBL86754 | IODOQUINOL | 2.0 | 1 | 7.41 |
| CHEMBL12131 | CLOSANTEL | 2.0 | 1 | 7.36 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | — | 1 | 7.03 |
| CHEMBL388590 | BENZBROMARONE | 4.0 | 1 | 6.98 |
| CHEMBL47050 | PENFLURIDOL | 2.0 | 1 | 6.78 |
| CHEMBL1333953 | PHENYLMERCURIC ACETATE | — | 1 | 6.72 |
| CHEMBL3184339 | — | — | 1 | 6.69 |
| CHEMBL550348 | DEFERASIROX | 4.0 | 1 | 6.63 |
| CHEMBL79834 | SPIRAMIDE | 2.0 | 1 | 6.62 |
| CHEMBL3188653 | — | — | 1 | 6.60 |
| CHEMBL2355158 | — | — | 1 | 6.55 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 6.52 |
| CHEMBL417799 | SANGUINARIUM | 2.0 | 1 | 6.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL232201 | BENZIODARONE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL24944 | TRIBROMSALAN | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 1.47 | nM | 8.83 |
| CHEMBL50588 | EMETINE | IC50 | = | 2.28 | nM | 8.64 |
| CHEMBL3559830 | — | IC50 | = | 3.2 | nM | 8.49 |
| CHEMBL1375045 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5219790 | CETRIMIDE | IC50 | = | 5.17 | nM | 8.29 |
| CHEMBL290106 | BITHIONOL | IC50 | = | 8.67 | nM | 8.06 |
| CHEMBL1981438 | CLOFLUCARBAN | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL287542 | RAFOXANIDE | IC50 | = | 14.3 | nM | 7.84 |
| CHEMBL105442 | CI-1040 | IC50 | = | 17.1 | nM | 7.77 |
| CHEMBL81782 | — | IC50 | = | 17.21 | nM | 7.76 |
| CHEMBL2355417 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL2361697 | — | IC50 | = | 29.8 | nM | 7.53 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL1545634 | — | IC50 | = | 35.36 | nM | 7.45 |
| CHEMBL86754 | IODOQUINOL | IC50 | = | 38.7 | nM | 7.41 |
| CHEMBL12131 | CLOSANTEL | IC50 | = | 43.8 | nM | 7.36 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | IC50 | = | 94.1 | nM | 7.03 |
| CHEMBL388590 | BENZBROMARONE | IC50 | = | 105.3 | nM | 6.98 |
| CHEMBL47050 | PENFLURIDOL | IC50 | = | 167.5 | nM | 6.78 |
| CHEMBL1333953 | PHENYLMERCURIC ACETATE | IC50 | = | 192.0 | nM | 6.72 |
| CHEMBL3184339 | — | IC50 | = | 202.2 | nM | 6.69 |
| CHEMBL550348 | DEFERASIROX | IC50 | = | 232.76 | nM | 6.63 |
| CHEMBL79834 | SPIRAMIDE | IC50 | = | 241.58 | nM | 6.62 |
| CHEMBL3188653 | — | IC50 | = | 251.6 | nM | 6.60 |
| CHEMBL2355158 | — | IC50 | = | 279.5 | nM | 6.55 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 300.51 | nM | 6.52 |
| CHEMBL417799 | SANGUINARIUM | IC50 | = | 316.1 | nM | 6.50 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 332.09 | nM | 6.48 |
| CHEMBL1076347 | TRICLOCARBAN | IC50 | = | 334.6 | nM | 6.47 |
| CHEMBL178 | DAUNORUBICIN | IC50 | = | 337.6 | nM | 6.47 |
| CHEMBL51483 | GOSSYPOL | IC50 | = | 353.8 | nM | 6.45 |
| CHEMBL223448 | BROXYQUINOLINE | IC50 | = | 365.7 | nM | 6.44 |
| CHEMBL1450 | ATOVAQUONE | IC50 | = | 367.5 | nM | 6.43 |
| CHEMBL64894 | GENTIAN VIOLET | IC50 | = | 393.9 | nM | 6.41 |
| CHEMBL790 | CHLORHEXIDINE | IC50 | = | 438.6 | nM | 6.36 |
| CHEMBL2356978 | — | IC50 | = | 442.8 | nM | 6.35 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 472.85 | nM | 6.33 |
| CHEMBL497 | CLIOQUINOL | IC50 | = | 475.1 | nM | 6.32 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 498.82 | nM | 6.30 |
| CHEMBL1200596 | CHLOROXINE | IC50 | = | 495.2 | nM | 6.30 |
| CHEMBL1097558 | — | IC50 | = | 537.48 | nM | 6.27 |
| CHEMBL33845 | DICHLOROPHEN | IC50 | = | 546.4 | nM | 6.26 |
| CHEMBL939 | GEFITINIB | IC50 | = | 590.2 | nM | 6.23 |
| CHEMBL1571863 | ISOCONAZOLE | IC50 | = | 886.1 | nM | 6.05 |
| CHEMBL388676 | CAPTAN | IC50 | = | 902.6 | nM | 6.04 |
| CHEMBL334255 | CETYLPYRIDINIUM BROMIDE | IC50 | = | 934.0 | nM | 6.03 |
| CHEMBL125 | MILTEFOSINE | IC50 | = | 964.87 | nM | 6.02 |