Assay Detail
Functional
CHEMBL3562076
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Dry powder Dose response confirmation of uHTS inhibitor hits of the mitochondrial permeability transition pore via an absorbance. Mitochondrial Swelling.. (Class of assay: confirmatory)
101
Total Activities
100
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 101 | 4.87 | 6.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3561490 | — | — | 1 | 6.37 |
| CHEMBL1611438 | — | — | 1 | 6.16 |
| CHEMBL3560029 | — | — | 1 | 6.08 |
| CHEMBL3561163 | — | — | 1 | 6.02 |
| CHEMBL3560577 | — | — | 1 | 5.80 |
| CHEMBL1442924 | — | — | 1 | 5.76 |
| CHEMBL1331469 | — | — | 1 | 5.72 |
| CHEMBL3561283 | — | — | 1 | 5.65 |
| CHEMBL3560781 | — | — | 1 | 5.64 |
| CHEMBL1389776 | — | — | 1 | 5.64 |
| CHEMBL3561056 | — | — | 1 | 5.61 |
| CHEMBL3561865 | — | — | 1 | 5.48 |
| CHEMBL3559771 | — | — | 1 | 5.42 |
| CHEMBL3560986 | — | — | 1 | 5.34 |
| CHEMBL3561912 | — | — | 1 | 5.32 |
| CHEMBL3560869 | — | — | 1 | 5.30 |
| CHEMBL3560016 | — | — | 1 | 5.28 |
| CHEMBL3561476 | — | — | 1 | 5.22 |
| CHEMBL3561868 | — | — | 1 | 5.21 |
| CHEMBL3559746 | — | — | 1 | 5.20 |
| CHEMBL3560850 | — | — | 1 | 5.20 |
| CHEMBL3561680 | — | — | 1 | 5.00 |
| CHEMBL3560773 | — | — | 1 | 4.99 |
| CHEMBL3561905 | — | — | 1 | 4.98 |
| CHEMBL3561791 | — | — | 1 | 4.97 |
| CHEMBL3559859 | — | — | 1 | 4.87 |
| CHEMBL3561155 | — | — | 1 | 4.86 |
| CHEMBL3560025 | — | — | 1 | 4.86 |
| CHEMBL3561086 | — | — | 1 | 4.83 |
| CHEMBL3560345 | — | — | 1 | 4.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3561490 | — | IC50 | = | 423.0 | nM | 6.37 |
| CHEMBL1611438 | — | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL3560029 | — | IC50 | = | 830.0 | nM | 6.08 |
| CHEMBL3561163 | — | IC50 | = | 950.0 | nM | 6.02 |
| CHEMBL3560577 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL1442924 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1331469 | — | IC50 | = | 1920.0 | nM | 5.72 |
| CHEMBL3561283 | — | IC50 | = | 2237.0 | nM | 5.65 |
| CHEMBL1389776 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL3560781 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL3561056 | — | IC50 | = | 2440.0 | nM | 5.61 |
| CHEMBL3561865 | — | IC50 | = | 3310.0 | nM | 5.48 |
| CHEMBL3559771 | — | IC50 | = | 3839.0 | nM | 5.42 |
| CHEMBL3560986 | — | IC50 | = | 4610.0 | nM | 5.34 |
| CHEMBL3561912 | — | IC50 | = | 4740.0 | nM | 5.32 |
| CHEMBL3560869 | — | IC50 | = | 4960.0 | nM | 5.30 |
| CHEMBL3560016 | — | IC50 | = | 5280.0 | nM | 5.28 |
| CHEMBL3561476 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL3561868 | — | IC50 | = | 6130.0 | nM | 5.21 |
| CHEMBL3559746 | — | IC50 | = | 6350.0 | nM | 5.20 |
| CHEMBL3560850 | — | IC50 | = | 6340.0 | nM | 5.20 |
| CHEMBL3561680 | — | IC50 | = | 10120.0 | nM | 5.00 |
| CHEMBL3560773 | — | IC50 | = | 10340.0 | nM | 4.99 |
| CHEMBL3561905 | — | IC50 | = | 10410.0 | nM | 4.98 |
| CHEMBL3561791 | — | IC50 | = | 10730.0 | nM | 4.97 |
| CHEMBL3559859 | — | IC50 | = | 13510.0 | nM | 4.87 |
| CHEMBL3561155 | — | IC50 | = | 13750.0 | nM | 4.86 |
| CHEMBL3560025 | — | IC50 | = | 13930.0 | nM | 4.86 |
| CHEMBL3561086 | — | IC50 | = | 14930.0 | nM | 4.83 |
| CHEMBL3560065 | — | IC50 | = | 15050.0 | nM | 4.82 |
| CHEMBL3560345 | — | IC50 | = | 15020.0 | nM | 4.82 |
| CHEMBL3561688 | — | IC50 | = | 18230.0 | nM | 4.74 |
| CHEMBL3560985 | — | IC50 | = | 20100.0 | nM | 4.70 |
| CHEMBL3560722 | — | IC50 | = | 23300.0 | nM | 4.63 |
| CHEMBL3559910 | — | IC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL3559893 | — | IC50 | = | 25090.0 | nM | 4.60 |
| CHEMBL3561770 | — | IC50 | = | 27610.0 | nM | 4.56 |
| CHEMBL1500845 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL3560405 | — | IC50 | = | 39980.0 | nM | 4.40 |
| CHEMBL3559804 | — | IC50 | = | 40900.0 | nM | 4.39 |
| CHEMBL3560867 | — | IC50 | = | 44910.0 | nM | 4.35 |
| CHEMBL3560156 | — | IC50 | = | 46500.0 | nM | 4.33 |
| CHEMBL1713176 | — | IC50 | = | 47200.0 | nM | 4.33 |
| CHEMBL3561807 | — | IC50 | = | 47810.0 | nM | 4.32 |
| CHEMBL3559784 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3559862 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3559994 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3560019 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3560293 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3560326 | — | IC50 | = | 50000.0 | nM | 4.30 |