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Assay Detail

CHEMBL3579500

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimycobacterial activity against Mycobacterium bovis BCG
8
Total Activities
4
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mycobacterium tuberculosis
Confidence 1 — Organism
Curated By Autocuration

Target

Mycobacterium tuberculosis (CHEMBL360)
Type ORGANISM
Organism Mycobacterium tuberculosis

Publication

Aranciamycins I and J, Antimycobacterial Anthracyclines from an Australian Marine-Derived Streptomyces sp.
Khalil ZG, Raju R, Piggott AM, Salim AA, Blumenthal A, Capon RJ.
J Nat Prod (2015) 78 : 949 -952
PubMed 25789410 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.00 6.16
MIC 4 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3577667 2 6.16
CHEMBL3577666 2 6.10
CHEMBL3577668 2 5.96
CHEMBL1096602 ARANCIAMYCIN 2 5.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3577667 IC50 = 700.0 nM 6.16
CHEMBL3577666 IC50 = 800.0 nM 6.10
CHEMBL3577668 IC50 = 1100.0 nM 5.96
CHEMBL1096602 ARANCIAMYCIN IC50 = 1700.0 nM 5.77
CHEMBL3577666 MIC = 10000.0 nM -
CHEMBL3577667 MIC = 10000.0 nM -
CHEMBL3577668 MIC = 30000.0 nM -
CHEMBL1096602 ARANCIAMYCIN MIC = 30000.0 nM -