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Assay Detail

CHEMBL3592116

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human SK-MEL-2 cells assessed as inhibition of cell growth incubated for 48 hrs by SRB assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type SK-MEL-2
Confidence 1 — Organism
Curated By Autocuration

Target

SK-MEL-2 (CHEMBL614917)
Type CELL-LINE
Organism Homo sapiens

Publication

A new antibacterial octaketide and cytotoxic phenylethanoid glycosides from Pogostemon cablin (Blanco) Benth.
Kim KH, Beemelmanns C, Clardy J, Cao S.
Bioorg Med Chem Lett (2015) 25 : 2834 -2836
PubMed 25981688 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.47 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53463 DOXORUBICIN 4.0 1 9.00
CHEMBL3359821 1 5.35
CHEMBL444478 ACETOSIDE 2.0 1 5.07
CHEMBL3590257 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53463 DOXORUBICIN IC50 = 1.0 nM 9.00
CHEMBL3359821 IC50 = 4500.0 nM 5.35
CHEMBL444478 ACETOSIDE IC50 = 8520.0 nM 5.07
CHEMBL3590257 IC50 > 30000.0 nM -