Assay Detail
Binding
CHEMBL3598445
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Non-competitive inhibition of FucT-5 (unknown origin) using LacNAc as acceptor substrate
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5 (CHEMBL3146) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Beyond substrate analogues: new inhibitor chemotypes for glycosyltransferases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.01 | 5.01 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1170899 | — | — | 1 | 5.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1170899 | — | Ki | = | 9700.0 | nM | 5.01 |