Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3603664

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human H296R cell aggregates grown on matrigel incubated for 72 hrs by MTS assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type H296R
Confidence 1 — Organism
Curated By Autocuration

Publication

Design, Synthesis, and Biological Evaluation of a Series of Anthracene-9,10-dione Dioxime β-Catenin Pathway Inhibitors.
Soldi R, Horrigan SK, Cholody MW, Padia J, Sorna V, Bearss J, Gilcrease G, Bhalla K, Verma A, Vankayalapati H, Sharma S.
J Med Chem (2015) 58 : 5854 -5862
PubMed 26182238 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.47 7.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3601411 TEGAVIVINT 2.0 1 7.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3601411 TEGAVIVINT IC50 = 34.2 nM 7.47