Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3606614

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against mouse C3H10T1/2 cells after 24 hrs by FMCA
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Mus musculus
Cell Type C3H 10T1/2
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

ADMET (CHEMBL612558)
Type ADMET

Publication

Hedgehog inhibitors from Withania somnifera.
Yoneyama T, Arai MA, Sadhu SK, Ahmed F, Ishibashi M.
Bioorg Med Chem Lett (2015) 25 : 3541 -3544
PubMed 26169123 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.13 5.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2047410 1 5.39
CHEMBL517080 WITHAFERIN A 1.0 1 5.31
CHEMBL469945 1 4.68
CHEMBL3234469 1 -
CHEMBL1934585 1 -
CHEMBL1934583 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2047410 IC50 = 4100.0 nM 5.39
CHEMBL517080 WITHAFERIN A IC50 = 4900.0 nM 5.31
CHEMBL469945 IC50 = 21000.0 nM 4.68
CHEMBL3234469 IC50 > 25000.0 nM -
CHEMBL1934585 IC50 > 25000.0 nM -
CHEMBL1934583 IC50 > 25000.0 nM -