Assay Detail
Functional
CHEMBL3611927
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Antiviral activity against HIV
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human immunodeficiency virus |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Human immunodeficiency virus (CHEMBL613758) ↗| Type | ORGANISM |
| Organism | Human immunodeficiency virus |
Publication
Pyrroloaryls and pyrroloheteroaryls: Inhibitors of the HIV fusion/attachment, reverse transcriptase and integrase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.85 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL68274 | — | — | 1 | 5.52 |
| CHEMBL69767 | — | — | 1 | 4.70 |
| CHEMBL33236 | — | — | 1 | 4.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL68274 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL69767 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL33236 | — | IC50 | = | 46000.0 | nM | 4.34 |