Assay Detail
Functional
CHEMBL3618825
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Bovine viral diarrhea virus 1-NADL ATCC VR-534 infected in MDBK cells assessed as protection against virus-induced cytopathogenicity after 3 to 4 days by MTT assay
32
Total Activities
32
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Bovine viral diarrhea virus 1-NADL |
| Cell Type | MDBK |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis, cytotoxicity and antimicrobial activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 32 | 5.96 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | — | 1 | 5.96 |
| CHEMBL3617124 | — | — | 1 | - |
| CHEMBL3617112 | — | — | 1 | - |
| CHEMBL3617113 | — | — | 1 | - |
| CHEMBL1300890 | — | — | 1 | - |
| CHEMBL3617114 | — | — | 1 | - |
| CHEMBL601616 | — | — | 1 | - |
| CHEMBL3617115 | — | — | 1 | - |
| CHEMBL3617116 | — | — | 1 | - |
| CHEMBL3617117 | — | — | 1 | - |
| CHEMBL3617118 | — | — | 1 | - |
| CHEMBL3617119 | — | — | 1 | - |
| CHEMBL3617120 | — | — | 1 | - |
| CHEMBL3617121 | — | — | 1 | - |
| CHEMBL3617122 | — | — | 1 | - |
| CHEMBL3617109 | — | — | 1 | - |
| CHEMBL3617125 | — | — | 1 | - |
| CHEMBL3617126 | — | — | 1 | - |
| CHEMBL3617127 | — | — | 1 | - |
| CHEMBL3617210 | — | — | 1 | - |
| CHEMBL1370117 | — | — | 1 | - |
| CHEMBL3617211 | — | — | 1 | - |
| CHEMBL3617212 | — | — | 1 | - |
| CHEMBL3617213 | — | — | 1 | - |
| CHEMBL1404528 | — | — | 1 | - |
| CHEMBL3617214 | — | — | 1 | - |
| CHEMBL3617215 | — | — | 1 | - |
| CHEMBL3617216 | — | — | 1 | - |
| CHEMBL3087551 | — | — | 1 | - |
| CHEMBL3617123 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | EC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL3617115 | — | EC50 | > | 17000.0 | nM | - |
| CHEMBL3617122 | — | EC50 | > | 9000.0 | nM | - |
| CHEMBL3617121 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617120 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617119 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617118 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617117 | — | EC50 | > | 9500.0 | nM | - |
| CHEMBL3617116 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617109 | — | EC50 | > | 49000.0 | nM | - |
| CHEMBL601616 | — | EC50 | > | 19000.0 | nM | - |
| CHEMBL3617114 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL1300890 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617113 | — | EC50 | > | 11000.0 | nM | - |
| CHEMBL3617112 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617111 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617110 | — | EC50 | > | 41000.0 | nM | - |
| CHEMBL3617124 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL3617125 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617126 | — | EC50 | > | 64000.0 | nM | - |
| CHEMBL3617127 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617210 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1370117 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617211 | — | EC50 | > | 48000.0 | nM | - |
| CHEMBL3617212 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617213 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL1404528 | — | EC50 | > | 40000.0 | nM | - |
| CHEMBL3617214 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617215 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617216 | — | EC50 | > | 48000.0 | nM | - |
| CHEMBL3087551 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3617123 | — | EC50 | > | 52000.0 | nM | - |