Assay Detail
Binding
CHEMBL3626243
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of COX1 (unknown origin) using arachidonic acid substrate by colorimetric assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Pentafluorosulfanyl-containing flufenamic acid analogs: Syntheses, properties and biological activities.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 5.21 | 5.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3623735 | — | — | 1 | 5.75 |
| CHEMBL3623738 | — | — | 1 | 4.66 |
| CHEMBL3623737 | — | — | 1 | - |
| CHEMBL3623736 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3623735 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL3623738 | — | IC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL3623737 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3623736 | — | IC50 | > | 100000.0 | nM | - |