Assay Detail
Binding
CHEMBL3626545
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]histamine from rat histamine H4 receptor expressed in HEK293T cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | HEK-293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Functional Profiling of 2-Aminopyrimidine Histamine H4 Receptor Modulators.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.91 | 7.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1915540 | ADRIFORANT | 2.0 | 1 | 7.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1915540 | ADRIFORANT | Ki | = | 12.3 | nM | 7.91 |