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Assay Detail

CHEMBL3626604

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to rat alpha1 adrenergic receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Adrenergic receptor alpha-1 (CHEMBL1907610)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Therapeutic Potential of 5-HT6 Receptor Agonists.
Karila D, Freret T, Bouet V, Boulouard M, Dallemagne P, Rochais C.
J Med Chem (2015) 58 : 7901 -7912
PubMed 26099069 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.52 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL365751 1 6.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL365751 Ki = 300.0 nM 6.52