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Assay Detail

CHEMBL3635776

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human plasmatic BChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured every 2 mins by Ellman's method
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Tissue Plasma
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cholinesterase (CHEMBL1914)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Tacrine-Trolox Hybrids: A Novel Class of Centrally Active, Nonhepatotoxic Multi-Target-Directed Ligands Exerting Anticholinesterase and Antioxidant Activities with Low In Vivo Toxicity.
Nepovimova E, Korabecny J, Dolezal R, Babkova K, Ondrejicek A, Jun D, Sepsova V, Horova A, Hrabinova M, Soukup O, Bukum N, Jost P, Muckova L, Kassa J, Malinak D, Andrs M, Kuca K.
J Med Chem (2015) 58 : 8985 -9003
PubMed 26503905 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 25 6.48 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3632988 1 7.70
CHEMBL3410951 1 7.22
CHEMBL95 TACRINE 4.0 1 7.10
CHEMBL3632987 1 7.10
CHEMBL3410952 1 7.10
CHEMBL3632990 1 7.05
CHEMBL3632991 1 6.89
CHEMBL3410955 1 6.89
CHEMBL3410956 1 6.80
CHEMBL3410954 1 6.72
CHEMBL3632626 1 6.54
CHEMBL3632992 1 6.40
CHEMBL3632848 1 6.40
CHEMBL3632994 1 6.27
CHEMBL3410953 1 6.25
CHEMBL3632847 1 6.21
CHEMBL3632850 1 6.16
CHEMBL3632993 1 6.16
CHEMBL3632849 1 6.16
CHEMBL3632989 1 6.11
CHEMBL3632846 1 5.89
CHEMBL3632851 1 5.82
CHEMBL292314 1 5.75
CHEMBL1256415 1 4.75
CHEMBL153 TROLOX 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3632988 IC50 = 20.0 nM 7.70
CHEMBL3410951 IC50 = 60.0 nM 7.22
CHEMBL95 TACRINE IC50 = 80.0 nM 7.10
CHEMBL3632987 IC50 = 80.0 nM 7.10
CHEMBL3410952 IC50 = 80.0 nM 7.10
CHEMBL3632990 IC50 = 90.0 nM 7.05
CHEMBL3632991 IC50 = 130.0 nM 6.89
CHEMBL3410955 IC50 = 130.0 nM 6.89
CHEMBL3410956 IC50 = 160.0 nM 6.80
CHEMBL3410954 IC50 = 190.0 nM 6.72
CHEMBL3632626 IC50 = 290.0 nM 6.54
CHEMBL3632992 IC50 = 400.0 nM 6.40
CHEMBL3632848 IC50 = 400.0 nM 6.40
CHEMBL3632994 IC50 = 540.0 nM 6.27
CHEMBL3410953 IC50 = 560.0 nM 6.25
CHEMBL3632847 IC50 = 620.0 nM 6.21
CHEMBL3632850 IC50 = 700.0 nM 6.16
CHEMBL3632993 IC50 = 700.0 nM 6.16
CHEMBL3632849 IC50 = 690.0 nM 6.16
CHEMBL3632989 IC50 = 770.0 nM 6.11
CHEMBL3632846 IC50 = 1300.0 nM 5.89
CHEMBL3632851 IC50 = 1530.0 nM 5.82
CHEMBL292314 IC50 = 1780.0 nM 5.75
CHEMBL1256415 IC50 = 17560.0 nM 4.75
CHEMBL153 TROLOX IC50 > 1000000.0 nM -