Assay Detail
Binding
CHEMBL3720850
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human JIK kinase domain (2 to 318 residues) expressed in baculovirus assessed as remaining ATP level incubated for 2 hrs by luciferase-luciferin coupled chemiluminescent kinase assay
98
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Serine/threonine-protein kinase TAO3 (CHEMBL5701) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Tao Kinase Modulators And Method Of Use
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 98 | 7.09 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3716849 | — | — | 1 | 7.30 |
| CHEMBL3716742 | — | — | 1 | 7.30 |
| CHEMBL3716597 | — | — | 1 | 7.30 |
| CHEMBL3717391 | — | — | 1 | 7.30 |
| CHEMBL3717287 | — | — | 1 | 7.30 |
| CHEMBL3716788 | — | — | 1 | 7.30 |
| CHEMBL3715872 | — | — | 1 | 7.30 |
| CHEMBL3718164 | — | — | 1 | 7.30 |
| CHEMBL3715589 | — | — | 1 | 7.30 |
| CHEMBL3716416 | — | — | 1 | 7.30 |
| CHEMBL3717713 | — | — | 1 | 7.30 |
| CHEMBL3715942 | — | — | 1 | 7.30 |
| CHEMBL3719286 | — | — | 1 | 7.30 |
| CHEMBL3717468 | — | — | 1 | 7.30 |
| CHEMBL3716774 | — | — | 1 | 7.30 |
| CHEMBL3718473 | — | — | 1 | 7.30 |
| CHEMBL3718940 | — | — | 1 | 7.30 |
| CHEMBL3718965 | — | — | 1 | 7.30 |
| CHEMBL3719051 | — | — | 1 | 7.30 |
| CHEMBL3718891 | — | — | 1 | 7.30 |
| CHEMBL3715362 | — | — | 1 | 7.30 |
| CHEMBL3715956 | — | — | 1 | 7.30 |
| CHEMBL3716318 | — | — | 1 | 7.30 |
| CHEMBL3717111 | — | — | 1 | 7.30 |
| CHEMBL3717584 | — | — | 1 | 7.30 |
| CHEMBL3718736 | — | — | 1 | 7.30 |
| CHEMBL3715005 | — | — | 1 | 7.30 |
| CHEMBL3718166 | — | — | 1 | 7.30 |
| CHEMBL3717484 | — | — | 1 | 7.30 |
| CHEMBL3717193 | — | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3716742 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717713 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716416 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715589 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718164 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715872 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716788 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717287 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717391 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716597 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717193 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715806 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717373 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715987 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3719326 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717452 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718066 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716968 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716744 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3719286 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718473 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717484 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718166 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715005 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718736 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717584 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717111 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716318 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715956 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718891 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3719051 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718965 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3718940 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716849 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3716774 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717468 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715942 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3715362 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL3717335 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3717761 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3714849 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3719165 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3715050 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3718499 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3715041 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3717643 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3717552 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3716567 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3716888 | — | IC50 | >= | 5000.0 | nM | - |
| CHEMBL3716192 | — | IC50 | >= | 5000.0 | nM | - |