Assay Detail
Functional
CHEMBL3738673
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Reovirus 1 ATCC VR- 214 infected in BHK21 cells assessed as protection against virus-induced cytopathic effect after 3 or 4 days by MTT assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mammalian orthoreovirus 1 |
| Cell Type | BHK-21 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 29 | 4.86 | 5.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | — | 1 | 5.72 |
| CHEMBL3735511 | — | — | 1 | 4.68 |
| CHEMBL3735224 | — | — | 1 | 4.17 |
| CHEMBL1940475 | — | — | 1 | - |
| CHEMBL1940472 | — | — | 1 | - |
| CHEMBL3735424 | — | — | 1 | - |
| CHEMBL3735466 | — | — | 1 | - |
| CHEMBL3735360 | — | — | 1 | - |
| CHEMBL3734943 | — | — | 1 | - |
| CHEMBL3735842 | — | — | 1 | - |
| CHEMBL3736008 | — | — | 1 | - |
| CHEMBL3735926 | — | — | 1 | - |
| CHEMBL3736028 | — | — | 1 | - |
| CHEMBL3735703 | — | — | 1 | - |
| CHEMBL3734816 | — | — | 1 | - |
| CHEMBL1940474 | — | — | 1 | - |
| CHEMBL3734942 | — | — | 1 | - |
| CHEMBL3734906 | — | — | 1 | - |
| CHEMBL3735971 | — | — | 1 | - |
| CHEMBL3735304 | — | — | 1 | - |
| CHEMBL3735041 | — | — | 1 | - |
| CHEMBL3735827 | — | — | 1 | - |
| CHEMBL3734995 | — | — | 1 | - |
| CHEMBL3735809 | — | — | 1 | - |
| CHEMBL3736323 | — | — | 1 | - |
| CHEMBL3735060 | — | — | 1 | - |
| CHEMBL3735070 | — | — | 1 | - |
| CHEMBL438605 | — | — | 1 | - |
| CHEMBL3735085 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL3735511 | — | EC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL3735224 | — | EC50 | = | 67000.0 | nM | 4.17 |
| CHEMBL1940475 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1940472 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735424 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735466 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735360 | — | EC50 | > | 71000.0 | nM | - |
| CHEMBL3734943 | — | EC50 | > | 45000.0 | nM | - |
| CHEMBL3735842 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3736008 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735926 | — | EC50 | > | 15000.0 | nM | - |
| CHEMBL3736028 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735703 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL3734816 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1940474 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3734942 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3734906 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735971 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735304 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735041 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735827 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3734995 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735809 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3736323 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735060 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735070 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL438605 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3735085 | — | EC50 | > | 100000.0 | nM | - |