Assay Detail
Binding
CHEMBL3744100
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to adenosine A3 receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transmembrane domain-containing protein TMIGD3 (CHEMBL3712907) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
New substituted 9-propyladenine derivatives as A2Aadenosine receptor antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.24 | 5.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL576447 | — | — | 1 | 5.50 |
| CHEMBL567012 | — | — | 1 | 4.97 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL576447 | — | Ki | = | 3200.0 | nM | 5.50 |
| CHEMBL567012 | — | Ki | = | 10800.0 | nM | 4.97 |