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Assay Detail

CHEMBL3745445

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human thrombin preincubated for 10 mins using Ac-FVR-AMC as substrate by chromogenic assay
6
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Prothrombin (CHEMBL204)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Molecular modeling studies, synthesis and biological evaluation of dabigatran analogues as thrombin inhibitors.
Dong MH, Chen HF, Ren YJ, Shao FM.
Bioorg Med Chem (2016) 24 : 73 -84
PubMed 26690913 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 8.43 8.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL539697 DABIGATRAN ETEXILATE 4.0 2 8.58
CHEMBL3740928 2 8.40
CHEMBL3741603 2 8.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL539697 DABIGATRAN ETEXILATE IC50 = 2.63 nM 8.58
CHEMBL539697 DABIGATRAN ETEXILATE IC50 = 2.61 nM 8.58
CHEMBL3740928 IC50 = 3.981 nM 8.40
CHEMBL3740928 IC50 = 3.95 nM 8.40
CHEMBL3741603 IC50 = 5.012 nM 8.30
CHEMBL3741603 IC50 = 4.96 nM 8.30