Assay Detail
ADMET
CHEMBL3749034
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of aeromonas proteolytica aminopeptidase using L-leucine-p-nitroanilide as substrate by spectrophotometry
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Vibrio proteolyticus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Development of a novel sulfonate ester-based prodrug strategy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.72 | 6.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL225164 | CLOXYQUIN | 2.0 | 1 | 6.72 |
| CHEMBL3746376 | — | — | 1 | - |
| CHEMBL3747198 | — | — | 1 | - |
| CHEMBL3747278 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL225164 | CLOXYQUIN | Ki | = | 190.0 | nM | 6.72 |
| CHEMBL3746376 | — | Ki | > | 100000.0 | nM | - |
| CHEMBL3747198 | — | Ki | > | 100000.0 | nM | - |
| CHEMBL3747278 | — | Ki | > | 100000.0 | nM | - |