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Assay Detail

CHEMBL3750740

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Suppression of NO production in LPS-induced mouse RAW264.7 cells by Griess assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type RAW264.7
Confidence 1 — Organism
Curated By Autocuration

Target

RAW264.7 (CHEMBL612557)
Type CELL-LINE
Organism Mus musculus

Publication

Hit-to-lead optimization of phenylsulfonyl hydrazides for a potent suppressor of PGE2 production: Synthesis, biological activity, and molecular docking study.
Kim M, Lee S, Park EB, Kim KJ, Lee HH, Shin JS, Fischer K, Koeberle A, Werz O, Lee KT, Lee JY.
Bioorg Med Chem Lett (2016) 26 : 94 -99
PubMed 26602278 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.16 8.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3746729 1 8.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3746729 IC50 = 6.9 nM 8.16