Assay Detail
Binding
CHEMBL3755032
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Binding affinity to ERbeta (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structural features underlying raloxifene's biophysical interaction with bone matrix.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.51 | 8.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL431698 | RALOXIFENE CORE | — | 1 | 8.64 |
| CHEMBL81 | RALOXIFENE | 4.0 | 1 | 8.37 |
| CHEMBL1189544 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL431698 | RALOXIFENE CORE | Ki | = | 2.3 | nM | 8.64 |
| CHEMBL81 | RALOXIFENE | Ki | = | 4.3 | nM | 8.37 |
| CHEMBL1189544 | — | Ki | > | 10000.0 | nM | - |