Assay Detail
Binding
CHEMBL3760692
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at delta-opioid receptor in mouse vas deferens
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Tissue | Vas deferens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Multitarget opioid ligands in pain relief: New players in an old game.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ke | 2 | - | - |
| Kd | 1 | 9.25 | 9.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3759292 | — | — | 1 | 9.25 |
| CHEMBL3758231 | — | — | 1 | - |
| CHEMBL3758257 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3759292 | — | Kd | = | 0.5623 | nM | 9.25 |
| CHEMBL3758231 | — | Ke | = | 2.4 | nM | - |
| CHEMBL3758257 | — | Ke | = | 0.175 | nM | - |