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Assay Detail

CHEMBL3768680

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human NCI-H1299 cells assessed as reduction in cell viability after 48 hrs by MTT assay
6
Total Activities
6
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type NCI-H1299
Confidence 1 — Organism
Curated By Autocuration

Target

NCI-H1299 (CHEMBL612255)
Type CELL-LINE
Organism Homo sapiens

Publication

Carbohydrate-based inducers of cellular stress for targeting cancer cells.
Ndombera FT, VanHecke GC, Nagi S, Ahn YH.
Bioorg Med Chem Lett (2016) 26 : 1452 -1456
PubMed 26832785 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.25 4.52
Activity 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3765259 1 4.52
CHEMBL71595 HYDROGEN PEROXIDE 4.0 1 4.22
CHEMBL3765134 1 4.12
CHEMBL3765516 1 4.12
CHEMBL1236821 XYLOSE 4.0 1 -
CHEMBL3764021 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3765259 IC50 = 30000.0 nM 4.52
CHEMBL71595 HYDROGEN PEROXIDE IC50 = 60000.0 nM 4.22
CHEMBL3765134 IC50 = 75000.0 nM 4.12
CHEMBL3765516 IC50 = 75000.0 nM 4.12
CHEMBL1236821 XYLOSE Activity - -
CHEMBL3764021 Activity - -