Assay Detail
Binding
CHEMBL3772167
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]-CP 55,940 from human CB2 receptor expressed in CHO cells by liquid scintillation counting method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Ligand-based homology modelling of the human CB2receptor SR144528 antagonist binding site: a computational approach to explore the 1,5-diaryl pyrazole scaffold
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.22 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL381791 | — | — | 1 | 9.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL381791 | — | Ki | = | 0.6 | nM | 9.22 |