Assay Detail
Binding
CHEMBL3777319
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Displacement of [3H]LSD from rat cloned 5-Hydroxytryptamine receptor 7 after 60 mins
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Tactical Approaches to Interconverting GPCR Agonists and Antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 8.40 | 9.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL225284 | — | — | 1 | 9.66 |
| CHEMBL224820 | — | — | 1 | 8.18 |
| CHEMBL225512 | — | — | 1 | 7.94 |
| CHEMBL222755 | — | — | 1 | 7.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL225284 | — | Ki | = | 0.22 | nM | 9.66 |
| CHEMBL224820 | — | Ki | = | 6.6 | nM | 8.18 |
| CHEMBL225512 | — | Ki | = | 11.4 | nM | 7.94 |
| CHEMBL222755 | — | Ki | = | 15.2 | nM | 7.82 |