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Assay Detail

CHEMBL3779753

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [125I]Tyr11-somatostatin-14 from somatostatin receptor in mouse AtT20 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Cell Type AtT20
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Somatostatin receptor (CHEMBL2111427)
Type PROTEIN FAMILY
Organism Mus musculus

Publication

Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Waszkielewicz AM, Gunia-Krzyżak A, Powroźnik B, Słoczyńska K, Pękala E, Walczak M, Bednarski M, Żesławska E, Nitek W, Marona H.
Bioorg Med Chem (2016) 24 : 1793 -1810
PubMed 26988801 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 10.13 10.13

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1823872 SOMATOSTATIN 3.0 1 10.13

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1823872 SOMATOSTATIN IC50 = 0.074 nM 10.13