Assay Detail
Binding
CHEMBL3783503
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Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assay
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 8 | 8.91 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3781437 | — | — | 1 | 9.40 |
| CHEMBL3781953 | — | — | 1 | 9.29 |
| CHEMBL3779969 | — | — | 1 | 9.22 |
| CHEMBL3781521 | — | — | 1 | 9.16 |
| CHEMBL3781158 | — | — | 1 | 9.06 |
| CHEMBL3779954 | — | — | 1 | 8.89 |
| CHEMBL3780748 | — | — | 1 | 8.20 |
| CHEMBL3780020 | — | — | 1 | 8.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3781437 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL3781953 | — | EC50 | = | 0.51 | nM | 9.29 |
| CHEMBL3779969 | — | EC50 | = | 0.6 | nM | 9.22 |
| CHEMBL3781521 | — | EC50 | = | 0.69 | nM | 9.16 |
| CHEMBL3781158 | — | EC50 | = | 0.88 | nM | 9.06 |
| CHEMBL3779954 | — | EC50 | = | 1.28 | nM | 8.89 |
| CHEMBL3780748 | — | EC50 | = | 6.36 | nM | 8.20 |
| CHEMBL3780020 | — | EC50 | = | 8.67 | nM | 8.06 |